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Erlotinib

Generic Name: Erlotinib

Brand Names: Tarceva

Erlotinib is an EGFR inhibitor for non-small cell lung cancer and pancreatic cancer.

OncologyEGFR Inhibitor

What It's Used For

Erlotinib is prescribed for:

  • Non-small cell lung cancer with EGFR mutations
  • Pancreatic cancer (with gemcitabine)
  • Oncology targeted therapy

First-generation EGFR tyrosine kinase inhibitor.

Side Effects

Common side effects:

  • Rash (acneiform)
  • Diarrhea
  • Loss of appetite
  • Fatigue
  • Nausea

Serious side effects:

  • Interstitial lung disease
  • Hepatotoxicity
  • GI perforation
  • Severe skin reactions

Additional Information

What is Erlotinib?

Erlotinib is an EGFR inhibitor used for EGFR mutation-positive lung cancer.

EGFR Testing Required

EGFR mutation testing is required before starting - most effective in patients with activating EGFR mutations.

Take on Empty Stomach

Should be taken at least 1 hour before or 2 hours after food.

Learn more at MedlinePlus.

Medical Disclaimer: This information is for educational purposes only and should not be considered medical advice. Always consult with your healthcare provider before starting, stopping, or changing any medication. Your doctor can provide personalized recommendations based on your specific health condition and medical history.

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